Biotransformation of Digitoxigenin by Cochliobolus lunatus

نویسندگان

  • Rodrigo M. Pádua
  • Alaíde B. Oliveira
  • José D. Souza Filho
  • Jacqueline A. Takahashi
  • Maurício de Abreu
  • Fernão C. Braga
چکیده

A reação de biotransformação da digitoxigenina (1) por Cochliobolus lunatus foi investigada. Foram realizados experimentos com duração de 4 dias, que resultaram no isolamento de quatro produtos, cujas estruturas químicas foram elucidadas como sendo 1β-hidroxidigitoxigenina (2), 7β-hidroxidigitoxigenina (3), 8β-hidroxidigitoxigenina (4) e digitoxigenona (5). A obtenção desses produtos nas condições empregadas nunca foi anteriormente descrita. A produção da substância 4 em uma reação de biotransformação também é inédita.

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تاریخ انتشار 2007